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MK-8745
An Aurora A kinase inhibitor
PHA-680632
An Aurora kinase inhibitor
AT9283
A broad spectrum kinase inhibitor
TAK-901
A non-selective inhibitor of Aurora kinases
CCT129202
ENMD-2076 L-(+)-Tartaric acid
ENMD-2076 L-(+)-Tartaric acid 是一种多靶点激酶抑制剂,对 Aurora A、Flt3、KDR/VEGFR2、Flt4/VEGFR3、FGFR1 的 IC50 为 1.86、14、58.2、15.9、92.7、70.8、56.4 nM , FGFR2, Src, PDGFRα, 分别。
MLN8054
An inhibitor of Aurora A kinase
JNJ-7706621
A dual inhibitor of CDKs and Aurora kinases
MLN8237 (Alisertib)
XL228
A tyrosine kinase inhibitor
AMG-900
A selective pan-Aurora kinase inhibitor
Aurora A Inhibitor I
A potent and selective inhibitor of Aurora A kinase
Phthalazinone pyrazole
Potent, selective inhibitor of Aurora kinase A
SNS-314 Mesylate
A pan-Aurora kinase inhibitor
ZM 447439
Selective inhibitor of Aurora B kinase