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THZ1
A covalent Cdk7 inhibitor
LEE011
A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
PHA-767491
A potent Cdc7 kinase inhibitor
SNS-032 (BMS-387032)
A Cdk2, Cdk7, and Cdk9 inhibitor
Roscovitine (Seliciclib,CYC202)
A potent inhibitor of cyclin-dependent kinase 2
Cdk4/6 Inhibitor IV
A cell-permeable inhibitor of Cdk4/6
NSC 693868
A selective inhibitor of Cdk1 and Cdk5
CDK4 inhibitor
An antiproliferative cyclin D1/Cdk4 inhibitor
LY2835219 free base
A dual inhibitor of Cdk4 and Cdk6
A-674563
An Akt inhibitor
LY2857785
A Cdk9 inhibitor
BS-181
A selective Cdk7 inhibitor
P276-00
P276-00 (P276-00) 是一种有效的细胞周期蛋白依赖性激酶 (CDK) 抑制剂,可抑制 CDK9-cyclinT1、CDK4-cyclin D1 和 CDK1-cyclinB,IC50 分别为 20 nM、63 nM 和 79 nM。 P276-00 (P276-00) 对顺铂耐药细胞具有抗肿瘤活性。
SB1317
A multi-kinase inhibitor
Ro 3306
An inhibitor of Cdk1