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AMD 3465
A CXCR4 receptor antagonist
AMD 3465 hexahydrobromide
AMG 487 S-enantiomer
AMG 487 S-enantiomer 是 AMG 487 的 S 型异构体。AMG 487 是趋化因子受体 CXCR3 的有效拮抗剂。
CXCR7 modulator 1
CXCR7 modulator 1 (compound 25) 是具有口服活性的、CXCR7 类肽调节剂,其 Ki 值为 9 nM。
NBI-74330
A CXCR3 antagonist
Promazine hydrochloride
Promazine (Romtiazin, Sinophenin) is an antagonist at types 1, 2, and 4 dopamine receptors, 5-HT receptor types 2A and 2C, muscarinic receptors 1 through 5, alpha(1)-receptors, and histamine H1-receptors with antipsychotic effects.
SB 225002
Selective CXCR2 antagonist
Pridopidine (ACR16)
Pridopidine (ACR16, ASP2314, FR310826) , a dopamine (DA) stabilizer, acts as an antagonist against sigma 1 receptor (S1R) and dopamine D2 receptor (D2R).
3-Methoxytyramine (3-O-methyl Dopamine)
3-Methoxytyramine (3-O-methyl Dopamine) 是一种众所周知的 3-羟基酪胺/多巴胺的细胞外代谢物,是一种神经调节剂。
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride)
A natural metabolite of dopamine
Nicotinamide N-oxide
A metabolite of nicotinamide
Molindone hydrochloride (EN-1733A)
A dopamine receptor antagonist
WZ811
CXCR4 antagonist
AZD-5069
A CXCR2 antagonist
Reparixin
An allosteric inhibitor of CXCR1 and CXCR2