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Valeroyl Salicylate
A selective, irreversible inhibitor of COX-1
Etoricoxib
A selective COX-2 inhibitor
Acemetacin
An NSAID
Rofecoxib
A COX-2 inhibitor
N-(4-acetamidophenyl)-Indomethacin amide
Potent and selective reversible inhibitor of COX-2
SC 236
A potent, selective COX-2 inhibitor
(+/-)-Sulfinpyrazone
An inhibitor of uric acid reabsorption
Diclofenac
双氯芬酸是一种有效的非选择性抗炎药,作为 COX 抑制剂,对人 COX-1 和 COX-2 在 CHO 细胞中的 IC50 分别为 4 和 1.3 nM ,对羊 COX-1 的 IC50 分别为 5.1 和 0.84 μM和 COX-2,分别。
ZLJ-6
Dual inhibitor of cyclooxygenase/5-lipoxygenase
Pranoprofen
An NSAID and COX-1 inhibitor
Sulindac sulfone
A metabolite of sulindac
FK 3311
Tenidap
A COX-1 selective NSAID
Oxaprozin
An NSAID and COX inhibitor
NS 398
A selective COX2 inhibitor