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Ningetinib Tosylate
A multi-kinase inhibitor
MK-8033 hydrochloride
MK8033盐酸盐是ATP竞争性c-Met/Ron双重抑制剂,对野生型c-Met的IC50为1 nM,对c-Met N1100Y的IC50为2.0 nM。
c-met-IN-1
c-met-IN-1 (compound 16) 是一种高效选择性的 c-Met 抑制剂,IC50 值为 1.1 nM,具有抗肿瘤活性。
c-Met inhibitor 1
c-Met inhibitor 1是c-Met信号通路抑制剂,可作用于胃癌,胰腺癌和恶性胶质瘤。
2'-O,4'-C-Methyleneuridine
2’-O,4’-C-Methyleneuridine (Compound 15a) 是一种双环核苷。
TAS-115 mesylate (TAS-115 methanesulfonate)
TAS-115
ML-345
An inhibitor of the insulin-degrading enzyme
Savolitinib
An inhibitor of c-Met
CEP-40783
NVP-BVU972
A Met kinase inhibitor
Altiratinib
A multiple kinase inhibitor
MK-2461
A c-MET inhibitor
PF-04217903 methanesulfonate
A c-Met inhibitor
Tivantinib (ARQ 197)