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Fluo-DHA(NBD荧光标记双氢青蒿素)
Fluo-DHA是一种由NBD基团标记的双氢青蒿素(DHA)荧光探针,主要用于青蒿素药理学研究
Licochalcone B
Licochalcone B (Lico B), extracted from Glycyrrhiza uralensis Fisch, induces the cell cycle arrest and apoptosis in human hepatoma cell HepG2. Licochalcone B specifically inhibits the NLRP3 inflammasome by disrupting NEK7‐NLRP3 interaction.
Demethylzeylasteral
A nortriterpenoid with diverse biological activities
Esculin
A coumarin with antioxidant and anti-inflammatory activities
Diosbulbin B
Diosbulbin B 是从 D. bulbifera L. 中分离得到的二萜内酯,具有抗肿瘤活性。Diosbulbin B 可引起肝损伤 。
Ginsenoside Rh3
Ginsenoside Rh3 是 Ginsenoside Rg5 的细菌代谢产物。
Ruxolitinib (INCB018424)
Ruxolitinib (INCB18424)作为一种抑制剂,能够抑制Janus相关激酶(JAKs)JAK1和JAK2, IC50 分别为 3.3 nM 和 2.8 nM,Ruxolitinib介导对造血和免疫功能重要的若干细胞因子和生长因子信号。
Bromelaine(BR,300u/mg)
A mixture of proteolytic enzymes
Pepsin(porcine stomach mucose)(USP,1:30000)
蛋白质结构分析
Poly(ethylene glycol) diacrylate (MW:2000)
2,2'-Disulfanediylbis(ethan-1-ol),50% in Water
2,5-Dioxopyrrolidin-1-yl 2-bromoacetate
4-(2-Methylthiazol-4-yl)phenol
Cucurbituril
N,N'-Diphenylethylenediamine