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E3连接酶配体5是雌激素相关受体α; (ERRα) 拮抗剂,IC50 为 0.04 和 2.8 μM 代表 ERRα;和 ERRγ;分别。
E3 ligase Ligand 5 is a ligand of E3 ligase, extracted from patent US 20160058872A1, Paragraph 0515. E3 ligase Ligand 5 can be used in PROTAC technology.
[1]. Crew, Andrew P, et al. IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE. US20160058872A1.
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