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Trapoxin A
Trapoxin A is a cyclotetrapeptide histone deacetylase (HDAC) inhibitor.
PCI-34051
A potent, selective HDAC8 inhibitor
Trichostatin A (TSA)
A potent, reversible inhibitor of histone deacetylases
EDO-S101
An HDAC inhibitor and DNA alkylating agent
BRD 4354
BRD4354是HDAC5和HDAC9适度抑制剂,其IC50值分别为0.85,1.88μM。
Tefinostat
Tefinostat (CHR-2845) 是一种单核细胞/巨噬细胞靶向的 HDAC 广谱抑制剂,通过细胞内酯酶人羧酸酯酶-1 (hCE-1) 切割成活性酸 CHR-2847。具有抗抗单核细胞系白血病活性。
CAY10591
A SIRT1 activator
Nanatinostat
Nanatinostat (CHR-3996) 是一种有效的,有口服活性、I 类选择性的组蛋白去乙酰化酶 (HDAC) 抑制剂,IC50 值为 8 nM。
Tucidinostat
An HDAC inhibitor
TCS HDAC6 20b
An HDAC6 inhibitor
Domatinostat
Domatinostat (4SC-202) is a selective class I HDAC inhibitor with IC50 of 1.20 μM, 1.12 μM, and 0.57 μM for HDAC1, HDAC2, and HDAC3, respectively. Also displays inhibitory activity against Lysine specific demethylase 1 (LSD1). Phase 1.
TMP195
A class IIa HDAC inhibitor
ACY-1083
ACY-1083是一种可渗透脑的选择性HDAC6抑制剂,IC50为3nM,ACY-1083对HDAC6的选择性比其他类别的HDAC亚型高260倍。ACY-1083可有效逆转化疗引起的周围神经病变。
SR-4370
An HDAC3 inhibitor
Tenovin-6 Hydrochloride
A small molecule activator of p53