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PLX7904
A RAF inhibitor
GDC-0879
An inhibitor of B-RafV600E
B-Raf IN 1
An inhibitor of B-RAF and C-RAF
B-Raf inhibitor 1
An inhibitor of Raf kinases
MLN 2480
An oral pan-Raf kinase inhibitor
GW5074
A potent inhibitor of Raf-1
SB590885
A potent inhibitor of B-Raf
B-Raf inhibitor
B-Raf inhibitor 是一种有效的双重 TGFβ-activated kinase 1 (TAK1) 和 mitogen-activated protein kinase kinase kinase 2 (MAP4K2) 抑制剂,IC50 分别为 41.1 nM 和 18.2 nM。
BRAF inhibitor
BRAF 抑制剂是从专利 WO/2011103196 A1 化合物 P-0850 中提取的 B-Raf 抑制剂。
Dabrafenib Mesylate (GSK-2118436)
A Raf kinase inhibitor
ZM336372
An activator of the Raf-1 signalling pathway
Vemurafenib (PLX4032, RG7204)
An inhibitor of mutant V600E and wild type B-Raf
Tarafenacin
Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM),选择性比 M2 受体高约 200 倍。
LY3009120
A pan-Raf and Raf dimer inhibitor
Regorafenib monohydrate
A multi-kinase inhibitor