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FIIN-3
An inhibitor of FGFRs
TG 100572 Hydrochloride
TG 100572 Hydrochloride 是多靶点激酶抑制剂,抑制受体酪氨酸激酶 (receptor tyrosine kinases) 和Src激酶 (Src kinases); 对VEGFR1,VEGFR2,FGFR1,FGFR2,PDGFRβ,Fgr,Fyn,Hck,Lck,Lyn,Src,Yes 的 IC50 值分别为2,7,2,16,13,5,0.5,6,0.1,0.4,1,0.2 nM。
AMI-1 free acid
AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor with IC50 of 3.0 μM and 8.8 μM for yeast Hmt1p and human PRMT1, respectively.
BGJ398
An FGFR inhibitor
PD 173074
Inhibitor of tyrosine kinase activity of fibroblast growth factor receptors
TSU-68 (SU6668,Orantinib)
An inhibitor of select receptor tyrosine kinases
BLU-554
A potent inhibitor of FGFR4
FGFR4-IN-1
An inhibitor of FGFR4
S49076
S49076 是一种新型、有效的 MET、AXL/MER 和 FGFR1/2/3 抑制剂,IC50 值低于 20 nM。
CH5183284 (Debio-1347)
An inhibitor of FGFR1, 2, and 3
NVP-BGJ398 phosphate
NVP-BGJ398 phosphate (BGJ-398 phosphate; NVP-BGJ398 phosphate) 是一种有效的 FGFR 家族抑制剂,对 FGFR1、FGFR2、FGFR3 和 FGFR4 的 IC50 分别为 0.9 nM、1.4 nM、1 nM 和 60 nM。
Dovitinib lactate (CHIR-258 lactate)
A multi-kinase inhibitor
Tyrosine kinase-IN-1
Tyrosinekinase-IN-1是多靶点的酪氨酸激酶抑制剂,抑制KDR,Flt-1,FGFR1和PDGFRα的IC50值分别为4,20,4,2nM。
SSR128129E
Erdafitinib
A pan-FGFR inhibitor