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L-689502
L-689502是一个有效的HIV-1蛋白酶(HIV-lprotease)抑制剂,其IC50值为1nM。
CCR5 antagonist 1
CCR5antagonist1是一个CCR5拮抗剂,能够抑制HIV病毒的复制来自专利WO2004054974A2。
PNU-103017
PNU-103017是一种HIV蛋白酶抑制剂。
Dolutegravir-d5
A neuropeptide with diverse biological activities
C16 Globotriaosylceramide-d9 (d18:1/16:0-d9)
BRD-K98645985
BRD-K98645985 是一类 12 元大环内酰胺,也是一种 BAF (Brg/Brahma-associated factors) 转录阻遏的抑制剂,EC50 为 ~2.37 µM。BRD-K98645985 结合 ARID1A 特异的 BAF 复合物,防止核小体定位,并有效逆转 HIV-1 潜伏期,并且无 T 细胞毒性。
Dolutegravir O-β-D-Glucuronide
A metabolite of dolutegravir
(±)-Efavirenz-d5
An internal standard for the quantification of efavirenz
Benanomicin A
A microbial metabolite with antifungal, fungicidal, and antiviral activities
Benanomicin B (formate)
Cobicistat-d8
Globotriaosylceramides (hydroxy) (porcine)
Globotriaosycleramides are glycosphingolipids found in mammalian cell membranes that are synthesized from lactosylceramides.
Cabotegravir-d5
Darunavir-d9
An internal standard for the quantification of darunavir
Tenofovir diphosphate triethylamine
Tenofovirdiphosphatetriethylamine(TFV-DPtriethylamine)是一种ATP竞争性的DNA聚合酶(DNApolymerases)抑制剂,且是1型HIV(HIV-1)逆转录酶(RT)的底物。