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A-71623
A-71623 是一种基于 CCK-4 的肽,是一种有效且高度选择性的 CCK-A 完全激动剂。
(3R,4R)-A2-32-01
(3R,4R)-A2-32-01 (compound 2),抗毒力药物,是一种特异性的酪蛋白溶解蛋白蛋白酶 (ClpP) 抑制剂,EC50 值为 4.5 μM,并显示出可耐受的细胞毒性。
(3S,4S)-A2-32-01
(3S,4S)-A2-32-01 是 (3R,4R)-A2-32-01 的活性较低的 S-对映体。(3R,4R)-A2-32-01 是一种抗毒力剂和特异性酪蛋白水解蛋白酶 (ClpP) 抑制剂。
(R)-DRF053 dihydrochloride
cdk/CK1 inhibitor,potent and ATP-competitive
Casein Kinase II Inhibitor IV Hydrochloride
CaseinKinaseIIInhibitorIVHydrochloride是表皮角质形成细胞分化的小分子诱导剂。
SR 27897
A nonpeptide CCK1 antagonist
SSTC3
SSTC3 是 casein 激酶1α (CK1α) 的激动剂(Kd = 32 nM),可抑制WNT 信号 (EC50 = 30 nM)。SSTC3 与其他类型的 WNT 抑制剂相比,具有极小的胃肠道毒性。
BioE-1115
BioE-1115 is a highly selective and potent dual inhibitor of PAS kinase (PASK) and casein kinase 2α (CK2α) with IC50 of ~4 nM and ~10 μM, respectively.
4,5,6,7-Tetrabromobenzimidazole
A selective inhibitor of CK2
WL 47 - dimer
High affinity caveolin-1 ligand
CK1-IN-1
CK1-IN-1 (PUN51207, Compound 1C) is an inhibitor of casein kinase 1 (CK1) with IC50 of 15 nM, 16 nM and 73 nM for CK1δ, CK1ε and p38α MAPK, respectively.
Casein Kinase 2 Substrate (trifluoroacetate salt)
A peptide substrate for CK2
β-Casomorphin, human TFA
β-Casomorphin,humanTFA(Humanβ-casomorphin7TFA)是一种阿片样肽,作为opioid受体激动剂。
TA 01
An inducer of cardiomyocyte differentiation
Tryptone
酪蛋白胰消化物