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Bay 11-7821
A selective and irreversible NF-κB inhibitor
Lenalidomide hemihydrate
An analog of thalidomide
Lenalidomide hydrochloride
CPI-1189
A benzamide
O-Methylviridicatin
An inhibitor of TNF-α-induced HIV replication
Maslinic Acid
A biologically active triterpene
AX-024 hydrochloride
An inhibitor of the CD3ε-Nck interaction
SD 0006
An inhibitor of p38α MAPK
Infliximab
Infliximab (Avakine) 是一种嵌合单克隆 IgG1 抗体,可特异性结合 TNF-α。
R-8507
An antagonist of TNF-α receptor signaling
TNF-α Antagonist
A peptidomimetic of the TNF-α receptor ligand binding site
Hispidol ((Z)-Hispidol)
Hispidol ((Z)-Hispidol) ((Z)-Hispidol ((Z)-Hispidol)) 是炎症性肠病的潜在治疗剂;抑制 TNF-α;诱导单核细胞与结肠上皮细胞的粘附,IC50 为 0.50 μM.
Ginsenoside Rk3
GinsenosideRk3存在于Panaxnotoginseng的根中。在HepG2细胞中GinsenosideRk3抑制TNF-α诱导的NF-κB转录活性,IC50值为14.24±1.30μM。
SPD304
A small-molecule inhibitor of TNFα activity
Cynaropicrin
A sesquiterpene lactone