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Dalfopristin (mesylate)
A streptogramin antibiotic
Tedizolid HCl
Oxazolidinone for gram-positive infections
N-Tetradecanoyl-DL-homoserine lactone
N-tetradecanoyl-DL-homoserine lactone is a member of the N-acyl-homoserine lactone family.
N-(3-Hydroxyoctanoyl)-DL-homoserine lactone
N-(3-Hydroxyoctanoyl)-DL-homoserine lactone 是 N-acyl-homoserine lactone 家族的成员。
MBX-4132
MBX-4132,一种称为恶二唑的化学类别的成员,通过与细菌核糖体结合来抑制反式翻译。
6-CFDA N-succinimidyl ester
The succinimidyl ester group is capable of spontaneously and irreversibly binding to free amines
Entadamide-A-β-D-glucopyranoside
Entadamide-A-β-D-吡喃葡萄糖苷是 Entada phaseoloides 种子中的主要成分之一。
Cephapirin Benzathine
Cephapirin Benzathine 是头孢匹林的苄星盐形式。
Oritavancin diphosphate (LY333328 diphosphate)
Oritavancin Diphosphate is an orally active glycopeptide antibiotic which is active against Gram-positive bacteria and also has antibacterial activity against multidrug-resistant Streptococcus pneumoniae.
Closthioamide
Closthioamide是细菌DNA促旋酶的一个有效抑制剂,其对Ec,MRSA,VRE,Mv的最小抑菌浓度分别是9.00μM,0.58μM,0.58μM和72.03μM。
PF 03709270 (ulopenem etzadroxil)
PF 03709270 (ulopenem etzadroxil) (PF-03709270) 是一种口服可用的酯类前药形式的 sulopenem,对大多数革兰氏阳性菌和革兰氏阴性菌具有广谱抗菌活性。
Taniborbactam
Taniborbactam是一种有效的β-lactamase抑制剂,对β-lactamase不同亚型SHV-5,KPC-2,VIM-2和AmpC的IC50值<100nM,对OXA-1的IC50值为0.1-1μM,可用于细菌感染的研究。
Flagelin 22(TFA) (Flagellin 22(TFA))
Cecropin A TFA
CecropinATFA是由37个氨基酸残基构成的线性抗菌肽,从Hyalaphoracecropiapupae得到,具有抗菌、抗炎和抗癌作用。
RNAIII-inhibiting peptide(TFA)
RNAIII-inhibitingpeptide(TFA)是一种有效的Staphylococcusaureus多肽抑制剂,在蜂窝组织炎、角膜炎、化脓性关节炎、骨肌炎和乳腺炎等疾病中有功效。