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STM2457
STM2457 是一种首创的,高效、选择性的,具有口服活性的 METTL3 抑制剂,其 IC50 为 16.9 nM.,可用于急性白血病的研究。
Tetrahydrouridine (THU)
A cytidine deaminase inhibitor
CM-579 trihydrochloride
CM-579 trihydrochloride 是一线的、可逆的,G9a 和DNA 甲基转移酶 (DNMT) 的双抑制剂,其IC50 值分别为 16 nM 和32 nM。在多种癌细胞中发挥有效活性作用。
K-TMZ
A DNA alkylating agent
DS-437
A dual inhibitor of PRMT5 and PRMT7
4-(Methylnitrosamino)-1-(3-pyridyl)-1-butanone
A tobacco-specific nitrosamine carcinogen
Bobcat 339
A cytosine derivative
Decitabine-15N4
A neuropeptide with diverse biological activities
5-Fluoro-2'-deoxycytidine
2'-Deoxy-5-fluorocytidine (5-fluoro-2(')-deoxycytidine, FCdR), a pyrimidine analog, is a DNA methyltransferase (DMNT) inhibitor currently in clinical trials for solid tumors.
5-Azacytidine
A DNA methyltransferase inhibitor
2',3',5'-triacetyl-5-Azacytidine
A prodrug form of 5-azacytidine
RG 108
DNA methyltransferase inhibitor
SGI-110
SGI-110 (SGI-110) 是第二代 DNA 甲基转移酶 (DNMT) 抑制剂,用于研究急性髓性白血病 (AML) 和骨髓增生异常综合征 (MDS)。
SW155246
A DNA methyltransferase 1 inhibitor
S-(5'-Adenosyl)-L-methionine (tosylate)
S-Adenosyl-L-methioninetosylate(S-Adenosylmethioninetosylate)是通过蛋氨酸腺苷转移酶的作用由蛋氨酸和ATP内源性生产的,是一种重要的具有口服活性的甲基供体。