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Parecoxib
A prodrug form of valdecoxib
Indobufen
Indobufen (Ibustrin, K 3920) is a reversible platelet aggregation inhibitor. Indobufen is a reversible inhibitor of platelet cyclooxygenase (Cox) activity and suppresses thromboxane synthesis.
Imrecoxib
Imrecoxib(BAP-909)艾瑞昔布是选择性环氧合酶 2 (COX-2) 抑制剂,IC50 值为 18 nM,也可以抑制 COX1 活性,IC50 值为 115 nM。Imrecoxib(BAP-909) 艾瑞昔布具有抗炎作用。
GW-406381
A NSAID and COX-2 inhibitor
Etoricoxib D4
Etoricoxib D4 (MK-0663 D4) 是 Etoricoxib 的氘代标记物。Etoricoxib 是一种非甾体抗炎剂,为可口服的、选择性的 COX-2 抑制剂,对人全血 COX-2 和 COX-1 的 IC50 值分别为 1.1 μM 和 116 μM。
Benzoylgomisin O
Benzoylgomisin O 是从 Schisandra rubriflora 中分离的化合物,对 15-LOX、COX-1、COX-2 酶有抑制作用,且具有抗炎活性。
[10]-Shogaol
A phenol with diverse biological activities
(R)-Ketorolac
(R)-Ketorolac 是 Ketorolac 的 R 型对应体,可有效阵痛,减少溃疡的发生。(R)-Ketorolac 对 COX 无作用。
Hexahydrocurcumin
A natural product and an active metabolite of curcumin
Nitroflurbiprofen (HCT 1206)
Nitroflurbiprofen (HCT 1206) 是一种环氧合酶 (COX) 抑制剂,具有提供一氧化氮 (NO) 的特性,可调节门脉高压性肝硬化大鼠肝内血管张力的增加。
FR-188582
FR-188582是高选择性的环氧合酶(COX-2)抑制剂,IC50值为17nM。
Propyphenazone (4-Isopropylantipyrine)
Propyphenazone(4-Isopropylantipyrine, Isopropyrine), an analgesic and antipyretic agent, is a selective cyclooxygenase-2 inhibitor with anti-inflammatory activity.
Inulicin (1-O-Acetylbritannilactone)
A sesquiterpene lactone with diverse biological activities
(-)-Catechin gallate ((-)-Catechin 3-gallate)
A polyphenol with diverse biological activities
Catechin ((+)-Catechin)
(+)-Catechin (Cianidanol, Catechinic acid, Catechuic acid) is an antioxidant flavonoid, occurring especially in woody plants as both (+)-catechin and (-)-epicatechin (cis) forms.