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Tonapofylline
Tonapofylline (BG 9928) 是一种具有口服活性和选择性 A1 腺苷受体拮抗剂,对人 A1 腺苷受体 (hA1) 的 Ki 为 7.4 nM,选择性高出 A2A 腺苷受体 915 倍,A2B 腺苷受体 12 倍,正在开发为治疗心力衰竭的药物。
Swertisin
A flavonoid C-glycoside with diverse biological activities
Adenosine 5'-monophosphate monohydrate
Adenosine 5'-monophosphate monohydrate (5'-Adenylic acid, 5'-AMP) is an activator of a class of protein kinases known as AMP-activated protein kinase (AMPK).
N6-Ethyladenosine
An adenosine A1 and A3 receptor agonist
LAS101057
A potent adenosine A2B receptor antagonist
CPI-444 (V81444)
An adenosine A2A receptor antagonist
A2B receptor antagonist 1
A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂,来自专利WO2009157938A1实例9B。
A2AR-agonist-1
An agonist of adenosine A2A receptor and inhibitor of ENT1
A2A receptor antagonist 1
A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。
Tecadenoson (CVT-510)
An adenosine A1 receptor agonist
PSB-1115 (potassium salt)
An adenosine A2B receptor antagonist
CAY10680
A dual inhibitor of monoamine oxidase B and adenosine A2A receptors
CAY10498
An A3 adenosine receptor antagonist
3-Propylxanthine
An adenosine receptor antagonist and PDE inhibitor
BAY-545